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SESSION A – WPU Ballroom |
Discussion Leader: Dr. Dennis Curran |
Time |
Presenter |
Title/Topic |
|
9:00 |
John
A. Porco, Jr., Professor of
Chemistry, BU; Director, CMLD-BU |
Center Talk: "Recent Progress at
the CMLD-BU." |
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|
9:45 |
Jeffrey
AubŽ, Professor of Medicinal
Chemistry, KU; Director, KU-CMLD |
Center Talk: KU-CMLD Advances in the Synthesis of
Heterocycles |
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|
10:30 |
Stuart
Schreiber, Professor of Chemical
Biology, Harvard BICMLD |
Center Talk: Linking Chemical Methodology and Library
Development |
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|
11:15 |
Peter
Wipf, Professor of Chemistry,
Pittsburgh; Director, UPCMLD |
Center Talk: From Chemical
Methodologies to Biological Tools |
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|
|
12:00 |
Working
Lunch/Administrative Meeting – WPU Dining Room A |
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|
Discussion Leaders: Dr. Grace Woo & Mr. Branko Mitasev |
2:00 |
Aaron
B. Beeler, Ph.D., Assistant
Director, CMLD-BU |
ÒMultidimensional Screening as a Tool for Reaction
DiscoveryÓ |
|
|
2:20 |
Stefan
Werner, Ph.D., Associate Director,
UPCMLD |
Structural Diversity as Design Element
in the Synthesis of Small Molecule Libraries |
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|
2:40 |
Sarathy Kesavan, Ph.D. |
Synthesis and Diversification of Functionalized
Indane Scaffolds |
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|
3:00 |
Jared
Shaw, Ph.D., BICMLD |
Synthesis
and Screening of Structurally Diverse Libraries |
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|
3:20 |
David
Vander Velde, Research Professor
of Medicinal Chemistry, KU |
Analytical and Computational Strategies at the
KU-CMLD |
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|
3:40 |
Jeffrey
L. Brodsky, Associate Professor of
Biological Sciences, Pittsburgh |
Biological Effects of Small Molecule Hsp70 Modulators |
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|
4:00 |
Steve Bryant, Ph.D., NIH/NLM/NCBI |
PubChem |
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|
|
4:20 |
WPU
Lounge: Poster Session |
Titles
listed in separate program; Food & drinks co-sponsored by UPCMLD &
FTI |
|
|
|
5:50 |
Robert
Armstrong, Ph.D., Vice President,
Eli Lilly & Company |
Lead
Generation Strategies at Lilly |
|
|
|
7:00 |
Dinner:
Grand Concourse, Station Square [pre-meeting
sign-up required; pickup in Holiday Inn Lobby @ 7 PM] |
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|
SESSION B – CSC Room 12 |
|
Time |
Presenter |
Title/Topic |
|
Discussion Leaders: Mr. Adam Hoye and Mr. Elliot Wang |
9:00 |
Eamon Comer, Ph.D. |
Skeletal
Diversity Derived from Stereoselective Additions to Nitro Olefins |
|
|
9:20 |
Richard
Larock , Professor of Chemistry,
Iowa State University |
Synthesis
of Heterocycles via Iodocyclization and Aryne Annulation |
||
|
9:40 |
Jon
Tunge, Assistant Professor of
Chemistry, KU |
Synthesis of Libraries via C-H Bond
Functionalization |
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|
10:00 |
Scott
Nelson, Associate Professor of
Chemistry, University of Pittsburgh |
Asymmetric
Claisen Rearrangements as Enabling Technology for Diversity-Oriented
Synthesis |
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|
10:20 |
Jamie Driscoll, Ph.D., NIH/NIMH |
The Small Molecule Repository |
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|
10:45 |
Dan
Kahne, Professor of Chemical
Biology, BICMLD |
Mastering
Carbohydrate Linkages for DOS |
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|
11:10 |
Donna Huryn, Ph.D., Scientific Advisor of the UPCMLD |
From Chemical
Methodologies to Biological Tools - Part II: Annotating the UP-CMLD Library |
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|
11:30 |
Izzat T. Raheem, Ph.D., BICMLD |
Enantioselective
Pictet-Spengler-type Cyclizations of Hydroxylactams: An Anion-Binding Model
to Explain Catalysis with Chiral Pyrrole-Thioureas |
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|
11:50 |
Mary Pat Happ, Ph.D., BICMLD |
Design
and Standardized Analysis of Primary Screening Data to Facilitate Follow-up
Chemistry |
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|
|
12:10 |
CLOSING
REMARKS |
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|
Dr. Stefan Werner |
12:30-1:00 |
Tour of UPCMLD Facilities |
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